Focus on Cellulose ethers

HPMC siv hauv cov tshuaj

HPMC siv hauv cov tshuaj

Hydroxypropyl methylcellulose (HPMC) yog ib qho cellulose derivative uas tau siv dav hauv kev lag luam tshuaj rau nws cov khoom tshwj xeeb.Nws yog semi-synthetic, dej-soluble, thiab non-ionic polymer uas siv tau los ua cov thickener, binder, film-forming agent, thiab lubricant.HPMC tau txais koob meej hauv cov tshuaj vim nws lub peev xwm los txhim kho qhov zoo thiab ruaj khov ntawm cov ntaub ntawv ntau npaum.

Khoom Kev piav qhia
Cov qauv tshuaj Semi-synthetic cellulose derivative
Molecular hnyav 10,000-1,500,000 g / mol
Degree ntawm kev hloov 0.9-1.7 Nws
Solubility Soluble nyob rau hauv dej thiab feem ntau organic solvents
pH stability Stable tshaj pH dav
Thermal stability Ruaj khov mus txog 200 ° C
viscosity Muaj peev xwm ntawm qis mus rau siab nyob ntawm qib
Particle loj 100 mesh (150 microns) los yog me dua
Qhov tshwm sim Dawb mus rau dawb hmoov los yog granules
tsw Tsis hnov ​​tsw
Saj Tasteless
Toxicity Non-toxic thiab non-irritating
Kev ua xua Tsis-allergenic
Neeg tsis noj nqaij / vegan Neeg tsis noj nqaij thiab vegan tus phooj ywg

 

Hauv tsab xov xwm no, peb yuav tham txog ntau yam kev siv ntawm HPMC hauv cov tshuaj hauv kev nthuav dav.

 

Tablet Formulation
HPMC feem ntau yog siv los ua cov ntaub ntawv hauv cov ntsiav tshuaj.Nws ua raws li kev sib khi tus neeg sawv cev los ntawm kev txhim kho cov khoom sib txuas ntawm cov ntsiav tshuaj granules, ua rau cov ntsiav tshuaj uas nyuaj thiab tsis tshua muaj kev sib tsoo.Tsis tas li ntawd, HPMC yog siv los ua disintegrant hauv cov ntsiav tshuaj formulations, txhawb cov ntsiav tshuaj disintegration thiab dissolution.HPMC tseem tuaj yeem siv los ua cov khoom siv txheej rau cov ntsiav tshuaj, uas pab tiv thaiv cov tshuaj los ntawm ib puag ncig, txhim kho kev ruaj ntseg, thiab tswj cov tshuaj tso tawm.

Capsule Formulation
HPMC yog siv los ua cov khoom siv tshuaj ntsiav hauv kev tsim khoom ntawm ob qho tib si tawv thiab mos gelatin capsules.Nws yog ib qho kev xaiv rau gelatin raws li nws yog neeg tsis noj nqaij, tsis muaj tshuaj lom, thiab tsis ua xua.HPMC capsules kuj tseem ruaj khov dua li cov gelatin capsules, vim lawv tsis raug kev txom nyem los ntawm kev sib txuas thiab tsis muaj xim.HPMC capsules tuaj yeem ua kom yaj hauv plab lossis cov hnyuv, nyob ntawm seb cov tshuaj yuav tsum tau tso tawm profile.

Ophthalmic Formulation
HPMC yog siv nyob rau hauv ophthalmic formulations raws li ib tug viscosity enhancer, muab lub sij hawm sib cuag nrog lub qhov muag thiab ntev tso tshuaj.Nws kuj yog siv los ua cov roj nplua nyeem, uas txo cov kev khaus khaus thiab txhim kho cov neeg mob kev nplij siab.

Tshuaj pleev ib ce
HPMC yog siv nyob rau hauv cov tshuaj pleev ib ce raws li ib tug thickening neeg sawv cev, muab viscosity thiab kev ntxhib los mos rau cream, gels, thiab lotions.Nws tseem tuaj yeem txhim kho kev ruaj ntseg ntawm kev tsim los ntawm kev txo cov syneresis thiab tiv thaiv kev sib cais theem.

Parenteral Formulation
HPMC yog siv nyob rau hauv parenteral formulations ua ib tug stabilizer thiab thickener.Nws pab tswj lub cev stability ntawm formulation, tiv thaiv particle aggregation thiab sedimentation.Nws kuj yog siv los ua tus neeg sawv cev ncua rau cov tshuaj tsis zoo soluble, kom ntseeg tau tias cov tshuaj sib txawv ntawm cov tshuaj hauv kev tsim.

Tswj Tso Tawm Formulation
HPMC feem ntau yog siv rau hauv kev txhim kho ntawm kev tswj kev tso tawm formulations.Nws tuaj yeem siv los ua cov khoom siv matrix, uas maj mam tso cov tshuaj dhau sijhawm.HPMC kuj tuaj yeem siv los hloov kho cov tshuaj tso tawm los ntawm kev hloov pauv cov ntsiab lus polymer, qhov hnyav molecular, thiab qib hloov pauv.

Mucoadhesive Formulation
HPMC yog siv nyob rau hauv mucoadhesive formulations vim nws muaj peev xwm mus ua raws li mucosal nto.Cov cuab yeej no tuaj yeem siv los txhim kho kev xa tshuaj mus rau qhov ncauj, qhov ntswg, thiab qhov chaw mos mucosa.HPMC kuj tseem tuaj yeem ncua sij hawm nyob hauv kev tsim, txhim kho kev nqus tshuaj thiab bioavailability.

Solubility Txhim Kho
HPMC tuaj yeem siv los txhim kho cov solubility ntawm cov tshuaj tsis zoo soluble.HPMC tsim complexes nrog cov tshuaj, ua rau nws solubility thiab dissolution tus nqi.Lub complexation yog nyob ntawm qhov hnyav molecular thiab degree ntawm kev hloov ntawm HPMC.

Rheology Hloov Kho
HPMC tuaj yeem siv los ua tus hloov kho rheology hauv ntau cov qauv.Nws tuaj yeem nce lossis txo qhov viscosity ntawm cov qauv, nyob ntawm qhov hnyav molecular thiab qib ntawm kev hloov ntawm HPMC.Cov cuab yeej no tuaj yeem siv los kho cov khoom ntws ntawm kev tsim, ua kom yooj yim rau kev tswj thiab txheej txheem.

Kev Kho Hniav Qhov ncauj
HPMC yog siv nyob rau hauv cov tshuaj kho qhov ncauj raws li ib tug thickener thiab binder.Nws tuaj yeem txhim kho qhov kev ntxhib los mos thiab viscosity ntawm cov tshuaj txhuam hniav,nrog rau txhim khu nws stability.Tsis tas li ntawd, HPMC tuaj yeem ua tus neeg sawv cev ua yeeb yaj kiab, muab kev tiv thaiv kev tiv thaiv ntawm cov hniav thiab cov pos hniav.

Suppository Formulation
HPMC yog siv nyob rau hauv suppository formulations raws li ib tug hauv paus khoom.Nws tuaj yeem muab kev tswj xyuas cov tshuaj tso tawm thiab txhim kho kev ua raws li tus neeg mob.HPMC suppositories tsis yog khaus thiab tsis muaj tshuaj lom, ua rau lawv tsim nyog siv rau hauv qhov chaw rhiab heev.

Kev kho mob daim ntawv
HPMC yog siv nyob rau hauv kev kho mob formulations raws li ib tug thickener thiab film-forming tus neeg sawv cev.Nws tuaj yeem pab tsim kev tiv thaiv kab mob ntawm lub qhov txhab, tiv thaiv kab mob thiab txhawb kev kho mob.HPMC tseem tuaj yeem txhim kho cov viscosity thiab kev ntxhib los mos ntawm cov ntaub qhwv lub qhov txhab, ua rau lawv yooj yim rau kev thov thiab tshem tawm.

Veterinary Formulation
HPMC yog siv nyob rau hauv veterinary formulations raws li ib tug binder thiab disintegrant nyob rau hauv cov ntsiav tshuaj thiab tsiav tshuaj.Nws tuaj yeem siv los ua cov thickener hauv gels thiab pastes.HPMC muaj kev nyab xeeb rau kev siv tsiaj thiab tsis muaj kev phom sij rau lawv txoj kev noj qab haus huv.

Excipient
HPMC feem ntau yog siv los ua ib qho ntxiv hauv cov tshuaj formulations.Nws yog ntau yam polymer uas tuaj yeem siv los hloov kho cov khoom ntawm kev tsim.HPMC yog inert thiab tsis muaj tshuaj lom, ua rau nws haum rau siv nyob rau hauv ntau hom ntau npaum li cas.

Hauv kev xaus, HPMC yog cov khoom siv dav siv polymer hauv kev lag luam tshuaj vim nws cov khoom tshwj xeeb.Nws yog siv los ua cov ntawv khi, disintegrant, txheej txheej, cov khoom siv tshuaj ntsiav, viscosity enhancer, lubricant, stabilizer, suspending agent, matrix material, mucoadhesive, solubility enhancer, rheology modifier, film-forming agent, and excipient.HPMC tsis muaj tshuaj lom, tsis ua xua, thiab muaj kev nyab xeeb siv rau tib neeg thiab tsiaj txhu.Nws versatility ua rau nws yog ib qho tseem ceeb nyob rau hauv ntau yam tshuaj formulations.

 

 


Post lub sij hawm: Mar-05-2023
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